LY2228820科研用抗肿瘤小分子靶向抑制剂

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DescriptionLY2228820 is a novel and potent inhibitor of p38 MAPK with IC50 of 7 nM.
Targetsp38α
Molecular Weight (MW)612.74
Formula

C24H29FN6.2CH4O3S

CAS No.862507-23-1, 862505-00-8 (free base), 862507-29-7 (HCl)
Chemical Name5-(2-tert-butyl-4-(4-fluorophenyl)-1H-imidazol-5-yl)-3-neopentyl-3H-imidazo[4,5-b]pyridin-2-amine dimethanesulfonate